24.04.30 (ȭ) 01:46

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üADC ҰK-̿, R&D
2024-03-19 05:50:40
üADC ҰK-̿, R&D
2024-03-19 05:50:40

5Ϻ 10ϱ ̱ȸ мȸ(AACR 2024)

ѡѹ̡̺񿤹̿ ü 鿪׾ ĺ Ұ

, ADC ü ӻ

[ϸ= ] ı ӻ Ȥ ǥϰ ִ ̿ žĺ ۷ι 뿡 . ̿ ü, ü๰ü(ADC) ۷ι ֽ Ʈ带 ݿ žĺ ⿡ . Ѿ, ѹ̾ǰ, ̺񿤹̿, ͹̿ ӻ ϸ غ ƴ.

19 迡 ̱ȸ мȸ(AACR 2024) 5Ϻ 5ϰ ̱ ̰ ֵȴ. ̱ȸ ̱ӻȸ(ASCO), ȸ(ESMO) Բ 3 ȸ зǸ ӻ, ӻ1 ׾Ͻž ĺ ʱ ӻ ַ Ұȴ.

ΰ Ÿϴ ü, Ȱ

̹ AACR 2024 ű Ÿϴ ü ĺ ӻ ȴ. ü ϳ ̸ Ÿϴ Ŭü Ư ׿ ߰ ־ ӻ ٴ 򰡸 ް ִ.

Ѿ ̿ó 鿪׾ ü ӻ 2 Ѵ.

ȸ ʷ Ǵ žĺ YH41723̴. YH41723 Ѿ ̹ÿ½þư 鿪׾ PD-L1 TIGIT ŸѴ. Ѿ ŰƮ, ɵ ȭ 鿪׾ Ÿϴ PD-L1 鿪 T NK ǥ鿡 ϼ TIGIT(T-cell iMMunoreceptor with immunoglobulin and ITIM domain) Ÿ ȿ شȭϰڴٴ ȹ̴. Ѿ ܿ ν, ũ, Ƽ, 渮 ۷ι TIGIT Ÿϴ ׾ ž ϰ ִ.

̿ܿ Ѿ ̺񿤹̿ 鿪׾ YH32367 ӻ ͷ Ѵ. YH32367 ֿ Ͽ Ǵ ̿Ŀ HER2 41BB ܹ ŸѴ. PD-L1 ϴ ϼ ֺ 鿪 41BB ȰȭDZ 41BB ۿ ּȭϸ ׾ ȿ Ÿ ˷ ִ.

ѹ̾ǰ PD-L1 41BB Ÿϴ BH3120 ӻ ǥѴ. BH3120 ѹ̾ǰ ÷ Žٵ ƴ. ̴ 鿪 Ȱȭϴ ÿ Ÿ ϼ ϴ ü ÷ ̴. ̹ мȸ PD-1 뿡 ׾ ó ȿ Ͽ ̴. BH3120 ϰѹ̾ǰ ӻ ֵϰ ܵ ӻ1 ǰ ִ.

ѹ̾ǰ EZH1/2 HM97662 ǥѴ. EZH2 EZH1 Ȱȭ ߵǴ ˷ ִ. ѹ̾ǰ EZH1 EZH2 ϴ EZH2 ܵ غ ȿ ִٴ HM97662 ϰ ִ.

̺񿤹̿ ̹ мȸ ο ü 鿪׾ ABL112 ABL407 ӻ ͷ Ѵ. žĺ 9 AACR 2024 ǥ Ǵ ű ̴. ABL112 ABL407 41BB ü ÷ ׷ٵ-T ƴ. ABL112 TIGIT, ABL407 鿪 ϴ LILRB4 ǥѴ.

鿪 õ 鿪 ÿ ϴ ٵ ü ʸø ǥѴ. ȸ PD-L1 õ 鿪 CD47 ÿ ۿ ϼ 鿪ȸ ؿ ׾ȿ ̴. ʸø 󵵿 Ű ʾ CD47 ü ۿ Ÿ ʴ ˷ ִ.


͹̿, ADC ü LCB36 ӻ ù

ü๰ü(ADC) ϰ ִ ͹̿ ̹ мȸ ADC ü LCB36 ӻ ó Ѵ. LCB36 CD20 CD22 Ÿϴ ADC. CD20̳ CD22 Ÿϴ Ŭü CD20XCD3 Ÿϴ ü ߵ CD20 CD22 Ÿϴ LCB36 ʴ.

CD20 CD22 ׾Ͽ Ǵ ˷ ͹̿ LCB36 B Ÿϴ ž ϰ ִ. ͹̿ 콺 𵨿 ༺ ȹ̴.

̿ܿ ͹̿ Ŭ 18.2 ǥ ADC LCB02A ȹ̴. Ŭ 18.2 ַ ĵϿ Ǵ ܹ, ֱ ADC ž о߿ ޺λϴ ǥ̴.

͹̿ TROP2 ǥϴ ADC LCB84 ӻ Ѵ. LCB84 12 ̱ ص(J&J) ȸ Ἶ 17 ޷( 2 2400) Ը ⿡ žĺ̴.

ӻ󿡼 LCB84 ̼ҸӶ ̷ε TROP2 ADC ๰ ϴ Ͽ ȿ ִ. ̼ҸӶ (ƮƮָ轺ĭ) ֿ ADC ̴.

TROP2 Į ȣ ȯ İ Ѵ. ش ܹ ϳ ϼ ϴ ๰׼ ִ ˷.

TROP2 ̿Ŀ ַ , Ҽ,  ַ Ȯεǰ ־ ͹̿ ߻ ֿ Ÿ ӻ ϰ ִ. ȭ 渮 Ʈε(ָĭ) ϴ.
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ֽż ݴ
  • 2024.03.19 06:59:00 |

    ڳ

    2Ⱓ ֵ ڳ~~~!!!

    0 5 0
ٺ Ϲݾ ǸŰ (2024 04)
౹ 31
ǰ ְ
ѽŻ÷(10) 3,500 2,500 1,000 3,009
޾(100) 24,000 23,000 1,000 23,200
Ʒγΰ(100) 30,000 28,000 2,000 28,500
īɾ(10g) 7,000 6,000 1,000 6,559
Ľõ򿬰(5g) 5,000 4,500 500 5,138
Ź(4) 5,000 4,000 1,000 4,438
ڶ(20) 6,000 6,000 0 6,000
(10) 6,000 4,500 1,500 5,071
Ժ(10) 4,000 3,500 500 3,712
ڱ׸(20) 5,000 4,500 500 4,717
ť(10) 3,000 2,500 500 2,990
Ȱť(1) 1,200 900 300 1,182
Ǯɾ(3.3ml) 26,000 23,000 3,000 24,250
޵𿬰(10g) 7,000 5,900 1,100 6,289
öŸ(34) 13,000 11,000 2,000 11,866
뽺ī(20g) 22,000 18,000 4,000 20,184
ġ(1) 1,000 1,000 0 1,000
ӽ÷(21) 10,000 8,500 1,500 9,205
ͺ(10) 3,500 3,000 500 3,196
ݿ(1ڽ) 3,000 3,000 0 3,000
׶÷糪ƮŸ(6) 8,000 7,000 1,000 7,524
߽Ÿ(120) 70,000 50,000 20,000 60,385
Źĸ(10ĸ) 3,000 2,000 1,000 2,989
Ÿ̾(120) 60,000 50,000 10,000 51,538
տ(60ĸ) 29,000 25,000 4,000 27,600
Ÿ̷ER(6) 3,000 2,500 500 2,750
ٿ(30g) 12,000 9,000 3,000 11,444
(120) 25,000 22,000 3,000 24,991
Ʒ(6) 4,000 3,000 1,000 3,262
ǽõĸ(270ĸ) 110,000 110,000 0 110,000
B(120) 70,000 70,000 0 70,000
׳(10) 3,000 2,500 500 2,778
6̺(10) 3,000 3,000 0 3,000
(60) 230,000 220,000 10,000 223,333
Ⱦ 12,000 10,000 2,000 10,143
̰źĸ(60ĸ) 35,000 30,000 5,000 33,231
Ųť(20) 5,500 4,500 1,000 4,903
λ絹÷(100) 35,000 32,000 3,000 33,297
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