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"TNF JAK鿪ȯ ߽ɿ 'ȭ' ִ"
ȣ 2020-10-08 06:20:40
"TNF JAK鿪ȯ ߽ɿ 'ȭ' ִ"
ȣ 2020-10-08 06:20:40

|ͺ| ѱȭ 鿪

'근' '', ٸ

Ȯ ȭ ׸
 
[ϸ=ȣ ] TNF- ڰ鿪ȯ з ȯ ๰̴.

Ƽ Ѿ TNF- ô߿, Ǽ, Ǽ پ Ȯ, ֿ ġɼ ڸҴ.

ִ. TNF- ȯ ϴ ȯڰ ϱ ̴.

ټ ȸ TNF- ߿ ߰ ߴŰ(JAK), ͷŲ(IL) ɼǵ ߴ.

̰ Ҷ ȭڴ ڰ鿪ȯ Ű÷̾ ϳ. ȸ TNF- '근(ŸʼƮ)' ϰ JAK ۽Ʈ Ŭ(First in class) ๰ '(ĽƼ)' ߴ.

۷ι ļ ๰ 'ƺνƼ' 㰡 â̴.

ϸ (44) ѱȭ 鿪(I&I, Inflammation&Immunology) , ڰ鿪ȯ ๰ Ʈ ô.

- Ұ ŹѴ.

ѱȭ I&Iθ Ѱϰ ִ. 2001 ѱȭ Ի ȯ, , ȣ, 鿪 پ ġ о߿ ð ׾ƿԴ.

پ ĿӼ ̲ 'ī࿧(丣ٽŸƾ, Ϸε)', '(Ȼ)', 'Ʈ()' ø ȭ ƽþ ͷμ 7 'ī(߸)' Ư㸸 ϱ⵵ ߴ.

-I&Iδ 2 ٽ ǰ ִ. ñϴ.

ǰ ѷ ȯڿ Ƿ鿡 ġ ϰ ִ. ǰ ġ ȿ ϰ ߴ.

2003 õ 근 16 ̻ 縦 ǰ̴. 근 Ƽ ġ з ٲٰ 򰡹޴ ๰, ش ġ о߿ ʷ TNF-̴.

鿪 TNF- ŭ, 근 ȯڱ 忡 ִ. Ư, źź ϰ ִٴ ū Ű ʹ.

Ƽ ο ġ з ๰̴. Ƽ ġ о߿ 汸 JAK , 2014 õ 2017 1ġ ޿ Ȯ ƴ.

Ƽ TNF-, ͷŲ پ ġɼ , ֻ ŭ ȯڵ 䰡 ߴ. ġ ä ȯڵ 並 ο ġ з ҷ ״ٰ 򰡹ް ִ.

- ๰ ġ Ѵ.  ִµ,  ϰ ֳ?

๰ ϱ⺸ٴ ȣ 迡 ִٰ . 근 Ƽ ϰ ϰ ִ ٸ.

근 ô߿ Ӹ ƴ϶ ޿ Ȯ ҾƯ߼(Ҿ ٰ , Ȯ强 Ҽ , Ǽ , ) ϰ ִ. Ư, ҾƯ߼ ȯڵ 䰡 ſ ȯڿ Ƿκ ȯ ޾Ҵ.

ݸ, Ƽ ˾缺忰 κп ϰ ִ.  Ȯǰ ִ ŭ, 근 ġ ְ δ ๰ 迡 ʴٰ Ѵ.

- ǷԴ JAK ó濡 庮 ϴ . ׷ Ƽ 忡 þ ִ ִٴ .

Ѵ. ѱ ġ(conventional therapy) ȣǴ ִ. ġ(early-treatment) ̷ Ѵٴ ٰŰ ǰ ġ ̿ ġῡ ӹ Ⱓ ̴. ְ ȯڵ ֻ δ㰨 ϳ .

׷  ʵη 汸 JAK ȯڵ鿡 ο Ƽ ġ ȯ ϴµ Ѵ. , Ƿ鿡Ե ġḦ ִ ȯ ϴ ū ϰ ִ.

-JAK ȭǰ ִ. ǰ Ӽ ϰ ƴ϶, Һ ŭ ׸ ӹϴ ̴.

Ƽ ȯ ȭ ȯ ־, Ȯ븦 鿪 ȯ ȯڵ鿡 Ƿ ֵ ̴. , Ƽ, ˾缺忰, Ǽ JAK ϰ ִ.

ȭڰ ϰ ִ JAK α׷ ̲ ǥ ๰̴. پ ȯڱ ȿ Ͱ Ǿ ִ. Ư, پ ȯڱ (RWD)  Ƿ ŷڸ ϰ ִ.

JAK 迭̱ ٸ ϰ ִ ŭ, ̷ ʹ  ִ Ͷ Ѵ.

-ڰ鿪ȯ ๰ Ǽ ġ ϴ°?

ڰ鿪ȯ ʿ ȯ, ʿϴ. Ư, ȯڵ ٸ ֻ縦 ϰ ϴ ѵ,  ϸ ȯڵ鿡 ġɼ ؿԴ.

ü Ǽ ǥϴ ๰̸ 근 , ֻ ʵø(Pre-filled Syringe) ܿ ȯڰ ϰ ڰֻ ֵ Ŭ(MyClic)̶ Ÿ Ұߴ. ǿ Ʈ Ű, ڰֻ ּȭ ֵ ֻ 90 ֵ ϱ ̺̽(E-Base) ⱸ ϰ ִ.

-ֱٿ JAK ִ.

ȭڴ Ӹ ƴ϶ پ JAK (JAK molecule) ∙ϸ ϰ ִ. , پ 鿪 Ű ȯ ġḦ ο ġ ϰ ִ. Ư Ƽȯ, ȭȯ, Ǻȯ ȯ ϰ ִ. ش ȯ ȯڵ鿡 ġɼ Ѵ.

-ݱ Ѱν θ ̲ 鼭 Ƿ, Ȥ شڵ 뿡 ־ٸ?

ȭڴ ȯڵ 䰡 ū ȯ Ǿǰ ∙ϱ ϰ ִ. ѱ ̷ Ͽ ȯڵ鿡 ġ ϰ ּ ϰ ִ.

׷ ž(first-in-class) ο ๰ , 㰡, ޿ ϴ ̴. ̷ ؼϱ Ƿ, ΰ پ ذڵ ϴ ȯ ޴ ȯڵ鿡  ϸ Ǿǰ ټ ϰ ִ.
ȣ (unkindfish@dailypharm.com) ٸ
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뺸 ϰ ̵ ̿ Ǵ ֽϴ.

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    弳 , Ӿ

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    Ÿ ID Ȥ г ϴ

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    ʴ

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    Խù б

  • û ִ

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    Ÿ ʻ ħϰų ϴ

    翡 ̿ (Ÿ ID, йȣ )

  • ̻ Ϻ ׿ ̿ 縦 , Ρ ó ֽϴ.

    õ ̴ ҹ Ǵܵǰų ϸ 񽺿 ٶ ʴٰ ǴܵǴ ġ ϰڽϴ.

    رŸ ϸ ڿ ֽʽÿ. ּҴ dailypharm@dailypharm.comԴϴ.

ֽż ݴ
ٺ Ϲݾ ǸŰ (2024 04)
౹ 31
ǰ ְ
ѽŻ÷(10) 3,500 2,500 1,000 3,009
޾(100) 24,000 23,000 1,000 23,200
Ʒγΰ(100) 30,000 28,000 2,000 28,500
īɾ(10g) 7,000 6,000 1,000 6,559
Ľõ򿬰(5g) 5,000 4,500 500 5,138
Ź(4) 5,000 4,000 1,000 4,438
ڶ(20) 6,000 6,000 0 6,000
(10) 6,000 4,500 1,500 5,071
Ժ(10) 4,000 3,500 500 3,712
ڱ׸(20) 5,000 4,500 500 4,717
ť(10) 3,000 2,500 500 2,990
Ȱť(1) 1,200 900 300 1,182
Ǯɾ(3.3ml) 26,000 23,000 3,000 24,250
޵𿬰(10g) 7,000 5,900 1,100 6,289
öŸ(34) 13,000 11,000 2,000 11,866
뽺ī(20g) 22,000 18,000 4,000 20,184
ġ(1) 1,000 1,000 0 1,000
ӽ÷(21) 10,000 8,500 1,500 9,205
ͺ(10) 3,500 3,000 500 3,196
ݿ(1ڽ) 3,000 3,000 0 3,000
׶÷糪ƮŸ(6) 8,000 7,000 1,000 7,524
߽Ÿ(120) 70,000 50,000 20,000 60,385
Źĸ(10ĸ) 3,000 2,000 1,000 2,989
Ÿ̾(120) 60,000 50,000 10,000 51,538
տ(60ĸ) 29,000 25,000 4,000 27,600
Ÿ̷ER(6) 3,000 2,500 500 2,750
ٿ(30g) 12,000 9,000 3,000 11,444
(120) 25,000 22,000 3,000 24,991
Ʒ(6) 4,000 3,000 1,000 3,262
ǽõĸ(270ĸ) 110,000 110,000 0 110,000
B(120) 70,000 70,000 0 70,000
׳(10) 3,000 2,500 500 2,778
6̺(10) 3,000 3,000 0 3,000
(60) 230,000 220,000 10,000 223,333
Ⱦ 12,000 10,000 2,000 10,143
̰źĸ(60ĸ) 35,000 30,000 5,000 33,231
Ųť(20) 5,500 4,500 1,000 4,903
λ絹÷(100) 35,000 32,000 3,000 33,297
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